Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5227441 | Tetrahedron | 2009 | 7 Pages |
Abstract
Efficient reaction conditions have been developed to prepare highly functionalized chiral pyranosido-pyrimidine by regioselective alkylation of the pyranoside ring and palladium-catalyzed cross-coupling reaction on the pyrimidine ring under microwave activation. Such scaffold contains three different functions suitable for selective derivatization and could find applications in the design of peptidomimetics.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Issa Samb, Nadia Pellegrini-Moïse, Sandrine Lamandé-Langle, Yves Chapleur,