PS-IIDQ: a supported coupling reagent for efficient and general amide bond formation

Article ID	Journal	Published Year	Pages	File Type
5229613	Tetrahedron	2007	17 Pages	PDF

Keywords

EDC O-(7-azabenzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate PyAOP Immobilized reagent MTBD NMM BOP HOAt TBTU HOBt DCC EEDQ 4-dimethylaminopyridine DMAP SPE DCE DMA THF dimethylacetamide DMF DCM 1-Ethyl-3-(3-dimethylaminopropyl)-carbodiimide 1-hydroxy-7-azabenzotriazole DMSO N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline N,N-dimethylformamide N,N-diisopropylethylamine Amide Tetrahydrofuran triethylamine Amide bond formation Amidation Microporous dimethyl-sulfoxide Dichloroethane Dichloromethane Parallel synthesis DIPEA HATU coupling reagent Polymer-supported reagent Polystyrene TEA

Related Topics

Physical Sciences and Engineering Chemistry Organic Chemistry

PS-IIDQ: a supported coupling reagent for efficient and general amide bond formation

Authors

Eric Valeur, Mark Bradley,