Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5262521 | Tetrahedron Letters | 2015 | 4 Pages |
Abstract
A highly efficient Rh(III)-catalyzed direct C-H arylation of indoles with aryl boronic acids under mild conditions has been developed. The methodology features wide substrate scope and excellent functional group compatibility (34 examples, up to 99% yield). The arylated products can also be conveniently transformed into biologically active polycyclic indole derivatives.66
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Liang Wang, Xing Qu, Zhan Li, Wang-Ming Peng,