Article ID Journal Published Year Pages File Type
5262521 Tetrahedron Letters 2015 4 Pages PDF
Abstract
A highly efficient Rh(III)-catalyzed direct C-H arylation of indoles with aryl boronic acids under mild conditions has been developed. The methodology features wide substrate scope and excellent functional group compatibility (34 examples, up to 99% yield). The arylated products can also be conveniently transformed into biologically active polycyclic indole derivatives.66
Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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