| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5264925 | Tetrahedron Letters | 2012 | 4 Pages |
Abstract
A facile two-step sequence (9â10â1) of regioselective assembly of 3,4-dihydroisoquinoline derivatives 1 is reported. The halogen derivatives provide opportunity for Suzuki, Buchwald, and related coupling reactions useful for expanding the scaffold and lead optimization in drug discovery.
Related Topics
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Authors
Zhongli Gao, Larry Davis, Yulin Chiang, Randall Munson, James A. Hendrix,