Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5266296 | Tetrahedron Letters | 2012 | 4 Pages |
Abstract
A divergent strategy for the synthesis of 1-aryl- and 2-aryl-2-iminoimidazolidines is presented. Cyclization of N-Boc-Nâ²-aryl-Nâ²â²-(2-hydroxyethyl)guanidines in the presence of methanesulfonyl chloride and triethylamine or sodium hydride at 0 °C affords the corresponding 2-iminoimidazolidines in good yields.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Daniel H. O'Donovan, Isabel Rozas,