Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5266440 | Tetrahedron Letters | 2013 | 5 Pages |
Abstract
Herein, we demonstrate the versatility of the pipecolic linker for the structural diversification of secondary amines with potential CNS activity. The solid-phase methods elaborated involved N1-indole sulfonylation, nitroindole and nitroarene reduction, and microwave-assisted Buchwald-Hartwig N-arylation.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
PaweÅ Zajdel, Nicolas Masurier, Vittorio Canale, Pascal Verdie, Muriel Amblard, Maciej PawÅowski, Jean Martinez, Gilles Subra,