| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5267184 | Tetrahedron Letters | 2011 | 4 Pages |
Abstract
The first one-pot three-component coupling reaction of O,O-diethyl hydrogen phosphorodithioate, aldehydes, and aldimines affording 1,2,4-trisubstituted 1,3-thiazetidines is reported. The product is obtained in moderate to high yields (45-94%) and has excellent diastereoselectivity (90-96%) in favour of the cis isomer. Shorter reaction times, ambient temperature, operational simplicity, and high yields are the salient features of the present procedure.
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Authors
Ankita Rai, Lal Dhar S. Yadav,