Article ID Journal Published Year Pages File Type
5267882 Tetrahedron Letters 2015 6 Pages PDF
Abstract

A palladium-catalyzed ortho-C-H-benzoxylation of 2-arylpyridines using iodobenzene dibenzoates has been developed. The reaction employed the stable and easily accessible hypervalent iodine reagents as both benzoxylate source and oxidant which made the protocol simple and facile. It showed high regioselectivity and good functional group tolerance, and gave the mono-benzoxylation products in moderate to excellent yields.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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