Article ID Journal Published Year Pages File Type
5268763 Tetrahedron Letters 2012 4 Pages PDF
Abstract

An efficient method for the preparation of various imidazobenzothiazine and primidobenzothiazine derivatives from readily available 2-mercaptoimidazoles (thiouracils) and bromobenzyl bromides via a copper(I)-catalyzed one-pot cascade process has been developed. The reaction involves a SN2 process and an intramolecular C-N cross coupling cyclization.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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