| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5268992 | Tetrahedron Letters | 2010 | 5 Pages |
Abstract
Direct N-arylation of urea (5) with various arylboronic acids mediated by cupric acetate furnished BIRB796 and a range of N-substituted BIRB796 analogs in good to moderate yields in one step. Urea (5) was readily synthesized from commercially available compounds.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Zhulin Tan, Jinhua J. Song, Jonathan T. Reeves, Daniel R. Fandrick, Heewon Lee, Scot Campbell, Nathan K. Yee,