Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5269110 | Tetrahedron Letters | 2011 | 5 Pages |
Abstract
Oxidative Heck coupling of thiazole-4-carboxylates via palladium(II)-catalyzed C-H bond activation has been achieved in moderate to good yields. No ligand, and no acidic additive were used in the reaction. The results showed that this protocol tolerated a series of substitutions on the thiazole ring. A preliminary attempt of direct arylation with p-xylene via Pd(II)-catalyzed C-H bond activation has also been done.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Ziyuan Li, Ling Ma, Changhua Tang, Jinyi Xu, Xiaoming Wu, Hequan Yao,