Article ID Journal Published Year Pages File Type
5269568 Tetrahedron Letters 2011 4 Pages PDF
Abstract

A general method for the Hiyama coupling reaction between aryl halides and 2-trimethylsilylpyridine has been developed. These conditions have been successfully applied to the synthesis of bis-heteroaryl systems, a key disconnection for the pharmaceutical industry in the synthesis of drug-like molecules.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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