Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5269822 | Tetrahedron Letters | 2010 | 4 Pages |
Abstract
An efficient, practical and environmentally benign synthesis of 2-substituted benzothiazoles was developed through RuCl3-catalyzed oxidative condensation of 2-aminothiophenol with aldehyde in ionic liquid by using air as the oxidant. With this procedure, a series of 2-substituted benzothiazoles and benzothiazole/pyrimidine nucleoside hybrids with antimicrobial activities were efficiently prepared from easily accessible starting materials.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Xuesen Fan, Yangyang Wang, Yan He, Xinying Zhang, Jianji Wang,