Article ID Journal Published Year Pages File Type
5270477 Tetrahedron Letters 2014 5 Pages PDF
Abstract

A highly environmentally benign protocol for the synthesis of quinazolinones from anthranilamides and aldehydes via aerobic oxidation was developed in wet DMSO. This protocol is operationally simple, exhibits broad substrate scope, and does not need toxic metal catalysts and bases. In addition, the utility of this transformation was further demonstrated by converting the resulting quinazolinones into other useful products in the same-pot without their isolation.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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