Article ID Journal Published Year Pages File Type
5271446 Tetrahedron Letters 2010 4 Pages PDF
Abstract

Herein we report a general synthesis of 1,3-diarylsubstituted indazoles utilizing a two-step Suzuki cross-coupling/deprotection/N-arylation sequence. This procedure proceeds in excellent overall yield starting from the 3-iodo-N-Boc indazole derivative allowing for rapid access to these compounds.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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