Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5271446 | Tetrahedron Letters | 2010 | 4 Pages |
Abstract
Herein we report a general synthesis of 1,3-diarylsubstituted indazoles utilizing a two-step Suzuki cross-coupling/deprotection/N-arylation sequence. This procedure proceeds in excellent overall yield starting from the 3-iodo-N-Boc indazole derivative allowing for rapid access to these compounds.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
James M. Salovich, Craig W. Lindsley, Corey R. Hopkins,