| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5271827 | Tetrahedron Letters | 2010 | 5 Pages |
Abstract
The first total synthesis of hirtellanines A is described. The key transformations include (i) base-mediated regioselective pyran ring formation, (ii) one-pot sequential boronation and Suzuki-Miyaura cross-coupling, and (iii) a tandem acid-induced deprotection and subsequent tautomerizations.
Graphical abstractThe first total synthesis of hirtellanine A was achieved in a high overall yield via the regioselective Claisen rearrangement as the key reaction.Download full-size image
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Shu-Yan Zheng, Zheng-Wu Shen,