Article ID Journal Published Year Pages File Type
5271925 Tetrahedron Letters 2013 5 Pages PDF
Abstract

A general and efficient reaction of indole with oxalyl chloride and nucleophiles providing indole-3-glyoxyl derivatives has been developed in mild conditions. In the same fashion, the other reaction involved the addition of organic azides leading to the synthesis of indole-3-glyoxyl-1,2,3-triazoles, which proceeds smoothly generating the products in moderate to high yields.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry