Article ID Journal Published Year Pages File Type
5272768 Tetrahedron Letters 2009 5 Pages PDF
Abstract

N-Boc-activated sulfahydantoin can be seen as glycine enolate equivalent. It appeared as a convenient starting material for the stereocontrolled preparation of threonine homologues through an alkaline syn aldolization involving a Boc migration. The methodology allowed the one-pot preparation of constrained analogues of polyoxamic acid.

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Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry