| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5273425 | Tetrahedron Letters | 2012 | 4 Pages |
Abstract
A method for the diastereoselective synthesis of tetrahydroquinolines via a palladium-catalyzed Suzuki terminated Heck reaction is described. The reaction provides access to tetrahydroquinolines containing both quaternary and tertiary stereocenters. Ligand effects, a rationale for the high level of diastereoselectivity, and a mechanistic hypothesis are discussed.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Jonathan E. Wilson,