Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5273522 | Tetrahedron Letters | 2008 | 4 Pages |
Abstract
Our study demonstrated that 4-(4,6-dimethoxy-1,3,5-triazine-2-yl)-4-methyl-morpholinium chloride (DMTMM) is a versatile coupling reagent for the synthesis of sterically-hindered peptidomimetics. It is superior to HBTU/HOBt and CDMT in controlling racemization and N-arylation, respectively.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Wen-Chung Shieh, Zhuoliang Chen, Song Xue, Joe McKenna, Run-Ming Wang, Kapa Prasad, Oljan RepiÄ,