Article ID Journal Published Year Pages File Type
5273978 Tetrahedron Letters 2013 6 Pages PDF
Abstract

A palladium-catalyzed cross coupling of nitrogen bearing heterocyclic chloromethyl derivatives with aryl and heteroaryl boronic acids has been developed. In almost all cases, highly efficient cross-couplings were observed at ambient temperature, mitigating unwanted thermally induced side-reactions. The comprehensive substrate scope and respectable yields highlight the synthetic utility of this reaction.

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Physical Sciences and Engineering Chemistry Organic Chemistry
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