| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5274058 | Tetrahedron Letters | 2009 | 4 Pages |
Abstract
New non-hydrolyzable analogues of glucosinolates have been prepared. Myrosinase inhibition was observed with modified aglycon moieties, even bulky phenothiazine analogue 6 gave reasonable inhibition. The simplest structure 8 derived from dimethylaminoethanethiol has shown to be the most potent inhibitor with an IC50 of 3.32 μM.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Deimante Cerniauskaite, Estelle Gallienne, Henreta Karciauskaite, Andrea S.F. Farinha, Jolanta Rousseau, Sylvie Armand, Arnaud Tatibouët, Algirdas Sackus, Patrick Rollin,