Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5274717 | Tetrahedron Letters | 2012 | 5 Pages |
Abstract
Access to the 1,5-disubstituted-1H-1,2,4-triazole-3-carboxamide motif is quite laborious and requires forcing conditions to effect the cyclocondensation step. Herein, we report an efficient and mild one-pot protocol to access this substructure in good chemical yields with high regiocontrol.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Sébastien Degorce, Bénédicte Delouvrié, Paul R.J. Davey, Myriam Didelot, Hervé Germain, Craig S. Harris, Christine Lambert-van der Brempt, Honorine Lebraud, Gilles Ouvry,