| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5274942 | Tetrahedron Letters | 2007 | 6 Pages |
Abstract
We have discovered a new route to 3-acylated indolizine structures via iodine-mediated hydrative cyclization. Reaction mechanism is proposed for this novel transformation, which involves a 5-exo-dig iodocyclization, deprotonation, incorporation of another iodo group, deprotonation, and subsequent replacement of the diiodo group by H2O. Various 3-acylated indolizine derivatives were obtained using this mild procedure in good yields.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Ikyon Kim, Sun Gi Kim, Ji Young Kim, Ge Hyeong Lee,