Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5275530 | Tetrahedron Letters | 2007 | 5 Pages |
Abstract
Glycals undergo smooth coupling with β-enaminoketones and β-enaminoesters generated in situ from 1,3-dicarbonyl compounds and arylamines in the presence of 10 mol % of InCl3 in refluxing dichloroethane to produce oxa-aza bicyclononene scaffolds in excellent yields with high selectivity. The use of InCl3 makes this protocol simple, convenient and easy to scale-up.
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Authors
J.S. Yadav, B.V. Subba Reddy, M. Srinivas, Ch. Divyavani, A.C. Kunwar, Ch. Madavi,