Article ID Journal Published Year Pages File Type
5276097 Tetrahedron Letters 2007 5 Pages PDF
Abstract

A mild and efficient allylation/propargylation of indoles has been developed with high regioselectivity and excellent yields. In the presence of catalytic molecular iodine, various indoles could react with allylic/propargylic acetates smoothly at room temperature to exclusively provide C-3 alkylated products.

Graphical abstractA mild and efficient allylation/propargylation of indoles has been developed with high regioselectivities and excellent yields. In the presence of catalytic molecular iodine, various indoles could smoothly react with allylic/propargylic acetates at room temperature to exclusively provide C-3 alkylated products.Download full-size image

Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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