| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5276428 | Tetrahedron Letters | 2012 | 5 Pages |
Abstract
An efficient and versatile methodology for the preparation of valuable triazolyl aminoacyl (peptidyl) penicillins is described. Solid-phase Cu(I)-catalyzed Hüisgen 1,3-dipolar cycloaddition was used as the key step showing general applicability and excellent regioselectivity either with CuI or [Cu(CH3CN)4]PF6 as Cu(I) source.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Patricia G. Cornier, Dora B. Boggián, Ernesto G. Mata, Carina M.L. Delpiccolo,