| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5277219 | Tetrahedron Letters | 2007 | 4 Pages |
Abstract
An efficient synthesis of 2-bromo-3-aryloxybenzothiophene derivatives by a conjugate addition-elimination sequence of 2,3-dibromo benzothiophene dioxides with phenolic nucleophiles has been developed. These benzothiophene derivatives serve as important intermediates for the synthesis of SERM analogues.
Graphical abstractAn efficient synthesis of 2-bromo-3-aryloxybenzothiophene by a conjugate addition-elimination sequence of 2,3-dibromo benzothiophene dioxides with phenolic nucleophiles has been developed.Download full-size image
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Fuyao Zhang, David Mitchell, Patrick Pollock, Tony Y. Zhang,