| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5278069 | Tetrahedron Letters | 2010 | 4 Pages |
Abstract
Aldehyde, homoallylic amine and arene undergo smooth cyclization in the presence of BF3·OEt2 to afford 4-arylpiperidines in good yields and with high trans-selectivity. This is the first report on the preparation of 4-arylpiperidines via aza-Prins-Friedel-Crafts reaction.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
J.S. Yadav, B.V. Subba Reddy, K. Ramesh, G.G.K.S. Narayana Kumar, René Grée,