Article ID Journal Published Year Pages File Type
5279388 Tetrahedron Letters 2006 5 Pages PDF
Abstract

A new family of pyrazole and bi-pyrazole phosphine ligands are reported that perform efficiently in the Pd-catalyzed amination reaction. Of the ligands screened, ligand 1 emerged as the most compatible for couplings involving both primary and secondary amines with typical yields of 84-99%.

Graphical abstractWe have prepared a new family of pyrazole and bi-pyrazole phosphine ligands that perform efficiently in the Pd-catalyzed amination reaction. Of the ligands screened, ligand 1 is the most compatible for couplings involving both primary and secondary amines with typical yields of 84-99%.Download full-size image

Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
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