Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5286749 | Tetrahedron Letters | 2005 | 4 Pages |
Abstract
The tin hydride-mediated cyclizations of a number of sulfides and sulfones under mild, neutral conditions, have been investigated accompanied by some amount of β-scission product for sulfides. The sulfides were derived from 4-mercaptoquinolone and 2-bromobenzyl bromides by phase transfer catalyzed reaction and the corresponding sulfones were prepared by treatment of the sulfides with m-CPBA at room temperature. The sulfides and the corresponding sulfones were then reacted with nBu3SnH-AIBN to give regioselective quinolone-annulated sulfur heterocycles.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
K.C. Majumdar, P.P. Mukhopadhyay, A. Biswas,