| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 5289243 | Tetrahedron Letters | 2006 | 4 Pages |
Abstract
A short, efficient synthesis of 4â³-(R or S)-4â³-deoxy-4â³-amino-4â³-C substituted avermectin B1 and 4â²-(R or S)-4â²-deoxy-4â²-amino-4â²-C substituted avermectin B1 monosaccharide 3 and 4 has been developed through the nucleophilic addition of an organometallic reagent to an intermediate phenylsulfinimide 7. These new derivatives of avermectin B1 exhibited potent, broad spectrum insecticidal activity.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Emmanuel Lamy, Patrick Lüthi, Clotilde Paturel, Tammo Winkler, Pierre M.J. Jung,