Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
7797587 | European Journal of Medicinal Chemistry | 2017 | 14 Pages |
Abstract
251Eight series of pyrrolo[2,3-b]pyridine and pyrrolo[2, 3-d]pyrimidine derivatives bearing pyridazinone moiety were designed, synthesized. Moreover, antitumor activity, enzyme-based selectivity, AO staining, Annexin V/PI staining and docking study were carried out.
Related Topics
Physical Sciences and Engineering
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Authors
Lin Xiao Wang, Xiaobo Liu, Shan Xu, Qidong Tang, Yongli Duan, Zhen Xiao, Jia Zhi, Liwen Jiang, Pengwu Zheng, Wufu Zhu,