Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
7798648 | European Journal of Medicinal Chemistry | 2016 | 8 Pages |
Keywords
NTDconcentration for 50% growth inhibitionTbNTRnifurtimox (4-(5-nitrofurfurylindenamino)-3-methylthio-morpholine-1,1-dioxide)benznidazole (N-benzyl-2-(2-nitro-1H-imidazol-1-yl)acetamide)T. bruceiT. cruziNfxType I nitroreductaseNTRCYP51Trypanosoma bruceiBNZIC50SARneglected tropical diseasesTrypanosoma cruziHuman African trypanosomiasisStructure-activity relationshipsselectivity indexChagas diseaseAntitrypanosomal agentsLeishmaniaHAT
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Maria V. Papadopoulou, William D. Bloomer, Howard S. Rosenzweig, Shane R. Wilkinson, Joanna Szular, Marcel Kaiser,