Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
7798835 | European Journal of Medicinal Chemistry | 2016 | 12 Pages |
Abstract
A series of novel arylpiperazine 5-(4-fluorophenyl)-5-methylhydantoins (2-15) was investigated on 5-HT7, 5-HT1A and D2 receptors affinity. VS/docking, synthesis, radioligand binding and functional assays as well as metabolic stability studies were performed.312
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Authors
Katarzyna Kucwaj-Brysz, Dawid Warszycki, Sabina Podlewska, Jagna Witek, Karolina Witek, Andrea González Izquierdo, Grzegorz SataÅa, MarÃa I. Loza, Annamaria Lubelska, Gniewomir Latacz, Andrzej J. Bojarski, Marián Castro, Katarzyna KieÄ-Kononowicz,