Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
7800160 | European Journal of Medicinal Chemistry | 2015 | 11 Pages |
Abstract
A series of N-benzooxazol-5-yl-pyrazole-4-carboxamides were designed and synthesized as potent SQR inhibitors. One candidate (Ki = 11 nM) was successfully identified as the most potent synthetic SQR inhibitor so far.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Li Xiong, Xiao-Lei Zhu, Yan-Qing Shen, Wickramabahu Kandergama Wasala Mudiyanselage Wishwajith, Kui Li, Guang-Fu Yang,