| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 7803022 | European Journal of Medicinal Chemistry | 2011 | 6 Pages |
Abstract
⺠Synthesis of aldehyde and vinylsulfone proteasome inhibitors. ⺠Proteasome inhibitors conjugated to the melanin-targeting ligand to target melanoma. ⺠Influence on the cytotoxicity of the benzamide alkyl side chain length. ⺠Influence on the cytotoxicity of the composition of the amino acid sequence. ⺠Cytotoxicity persisted in the presence of a melanin-targeting ligand.
Keywords
Related Topics
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Authors
Magali Vivier, Maryse Rapp, Marie-Josephe Galmier, Anne-Sophie Jarrousse, Elisabeth Miot-Noirault, Fernand Leal, Valérie Weber, Jacques Métin, Jacques Sauzière, Jean-Michel Chezal, Jean-Claude Madelmont,