Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
7803321 | European Journal of Medicinal Chemistry | 2011 | 8 Pages |
Abstract
⺠Synthesis of N-arylalkyl-2-(4-diphenylmethylpiperazin-1-yl)-4-hydroxybutyramide. ⺠Activity of murine GABA transport proteins GAT1-GAT4. ⺠The most active inhibitor with pKi = 4.96 in GAT1-binding assay.
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Authors
Katarzyna Kulig, Krzysztof WiÄckowski, Anna WiÄckowska, Justyna Gajda, BartÅomiej Pochwat, Georg C. Höfner, Klaus T. Wanner, Barbara Malawska,