Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Inhibitor; Sulfonamide; Carboxylic acid; Zinc-binding groups; Isoform-selective inhibitor
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Design, synthesis and biological evaluation of novel ureido benzenesulfonamides incorporating 1,3,5-triazine moieties as potent carbonic anhydrase IX inhibitors
Keywords: مهارکننده selective Isoform; Ureido benzenesulfonamides; 1,3,5-Triazine moiety; Carbonic anhydrase; Isoforms; Isoform-selective inhibitor; Cancer;
Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors
Keywords: مهارکننده selective Isoform; Triazene; Carbonic anhydrase; Isoforms; Isoform-selective inhibitor; Antiglaucoma agent;
Synthesis and biological evaluation of novel N,Nâ²-diaryl cyanoguanidines acting as potent and selective carbonic anhydrase II inhibitors
Keywords: مهارکننده selective Isoform; Cyanoguanidines; Carbonic anhydrase; Isoforms; Isoform-selective inhibitor; Antiglaucoma agent;
Synthesis and biological evaluation of novel aromatic and heterocyclic bis-sulfonamide Schiff bases as carbonic anhydrase I, II, VII and IX inhibitors
Keywords: مهارکننده selective Isoform; Bis-sulfonamide; Schiff base; Carbonic anhydrase; Isoform-selective inhibitor;
Inhibition of mammalian carbonic anhydrase isoforms I-XIV with a series of phenolic acid esters
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Phenol; Phenolic acid/ester; Isoform-selective inhibitor;
6-Triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrases IX and XII
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Sulfocoumarin; 1,4-Substituted 1,2,3-triazole; 1,5-Substituted 1,2,3-triazole; Click chemistry; Isoform-selective inhibitor; Tumor-associated carbonic anhydrase
Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: Identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Imine; Sulfonamide; Isoform-selective inhibitor; Tumor-associated enzymes;
Inhibition of human carbonic anhydrase isoforms I-XIV with sulfonamides incorporating fluorine and 1,3,5-triazine moieties
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Sulfonamide; 1,3,5-Triazine; Isoform-selective inhibitor;
7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Sulfocoumarin; Coumarin; Sulfonamide; Isoform-selective inhibitor;
Structural effect of phenyl ring compared to thiadiazole based adamantyl-sulfonamides on carbonic anhydrase inhibition
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Benzenesulfonamide; Adamantyl; X-ray crystallography; Isoform-selective inhibitor
Carbonic anhydrase inhibitors: Benzenesulfonamides incorporating cyanoacrylamide moieties are low nanomolar/subnanomolar inhibitors of the tumor-associated isoforms IX and XII
Keywords: مهارکننده selective Isoform; Sulfonamide; Carbonic anhydrase; Cyanoacrylamide; Isoform-selective inhibitor
5- and 6-Membered (thio)lactones are prodrug type carbonic anhydrase inhibitors
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Lactone; Thiolactone; Coumarin; Prodrug; Esterase activity; Isoform-selective inhibitor;
Phenylethynylbenzenesulfonamide regioisomers strongly and selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic isoforms I and II
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Isoforms I, II, IX, XII; Alkynylsulfonamide; Isoform-selective inhibitor; Antitumor lead;
Conformational variability of different sulfonamide inhibitors with thienyl-acetamido moieties attributes to differential binding in the active site of cytosolic human carbonic anhydrase isoforms
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Cytosolic isoforms; Sulfonamide; 2-Thienylacetamido tail; X-ray crystallography; Isoform-selective inhibitor
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Isoform IX, XII; Sulfonamide; 1,3,5-Triazine; X-ray crystallography; Isoform-selective inhibitor
7,8-Disubstituted- but not 6,7-disubstituted coumarins selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic ones I and II in the low nanomolar/subnanomolar range
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Tumor associated isoforms; Coumarin; Isoform-selective inhibitor; Fries rearrangement
Carbonic anhydrase inhibitors. Aromatic/heterocyclic sulfonamides incorporating phenacetyl, pyridylacetyl and thienylacetyl tails act as potent inhibitors of human mitochondrial isoforms VA and VB
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Cytosolic isoforms I and II; Mitochondrial isozymes VA and VB; Sulfonamide; Antiobesity; Isoform-selective inhibitor
Carbonic anhydrase inhibitors. Diazenylbenzenesulfonamides are potent and selective inhibitors of the tumor-associated isozymes IX and XII over the cytosolic isoforms I and II
Keywords: مهارکننده selective Isoform; Carbonic anhydrase; Tumor-associated isoforms; CA IX; CA XII; Isoform-selective inhibitor; Diazenylbenzenesulfonamides