| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 2006655 | Peptides | 2011 | 7 Pages |
Abstract
⺠A new tritiated endomorphin-2 analog was synthesized in which Pro2 is replaced by 2-aminocyclohexanecarboxylic acid. ⺠It shows high specific radioactivity, μ-opioid receptor affinity, selectivity and enzymatic resistance. ⺠It is a good tool to envisage the distribution of μ-opioid receptors by using receptor autoradiography. ⺠It may be more suitable than the parent ligand for receptor-ligand interaction and topographic studies.
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Authors
Attila Keresztes, Erika Birkás, Annamária Páhi, Géza Tóth, Lidia Bakota, Károly Gulya, Mária Szücs,