Potent inhibitors of human LAT1 (SLC7A5) transporter based on dithiazole and dithiazine compounds for development of anticancer drugs

Article ID	Journal	Published Year	Pages	File Type
5551966	Biochemical Pharmacology	2017	62 Pages	PDF

Keywords

CD98 2-amino-2-norbornanecarboxylic acid ADIC TX-100 dithioerythritol Pharmacological target ASCT2 C12E8 BCH SLC DTE mTOR octaethylene glycol monododecyl ether Triton X-100 solute carrier LAT blood brain barrier BBB Cancer Mechanism of inhibition mammalian target of rapamycin

Related Topics

Health Sciences Pharmacology, Toxicology and Pharmaceutical Science Pharmacology

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Potent inhibitors of human LAT1 (SLC7A5) transporter based on dithiazole and dithiazine compounds for development of anticancer drugs

Authors

Lara Napolitano, Mariafrancesca Scalise, Maria Koyioni, Panayiotis Koutentis, Marco Catto, Ivano Eberini, Chiara Parravicini, Luca Palazzolo, Leonardo Pisani, Michele Galluccio, Lara Console, Angelo Carotti, Cesare Indiveri,