| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 10586782 | Bioorganic & Medicinal Chemistry Letters | 2014 | 26 Pages |
Keywords
TC50EtOAcTHFDIEAHIADCMPBMCsHERGIC50ADMEDMFTFAHIV-1 EnvBioisostereBIFHeptad repeatN,N-diisopropylethylaminePd/CEthyl acetateTrifluoroacetic acidTetrahydrofuranHuman intestinal absorptionabsorption, distribution, metabolism, and excretionCNSdiisopropylethylaminedimethylformamideDichloromethaneBBBBlood–brain barrierperipheral blood mononuclear cellscentral nervous systemAntiviralEntry inhibitorDIPEAhalf-maximal inhibitory concentrationHATUhexafluorophosphatePalladium on carbonhuman ether-à-go-go-related genehigh-performance liquid chromatographyHPLC
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Marina Tuyishime, Matt Danish, Amy Princiotto, Marie K. Mankowski, Rae Lawrence, Henry-Georges Lombart, Kirill Esikov, Joel Berniac, Kuang Liang, Ji Jingjing, Roger G. Ptak, Navid Madani, Simon Cocklin,
