| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 10588587 | Bioorganic & Medicinal Chemistry Letters | 2011 | 4 Pages |
Abstract
The in vitro affinity of a series of N-substituted N-methyl-8-aminopentacyclo[5.4.0.02,6.03,10.05,9]undecanes for monoamine transporters DAT, NET, and SERT, is reported. Compound 12 was identified as a high affinity DAT ligand with excellent selectivity over the NET and SERT.
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Authors
Samuel D. Banister, Iman A. Moussa, Corinne Beinat, Aaron J. Reynolds, Paolo Schiavini, William T. Jorgensen, Michael Kassiou,