| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 10588747 | Bioorganic & Medicinal Chemistry Letters | 2011 | 4 Pages |
Abstract
Compound 2 was the culmination of SAR efforts from HTS lead 1. It has submicromolar potency in a HWB assay and efficacy in a CIA mouse model.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Timothy D. Cushing, Vijay Baichwal, Karen Berry, Roland Billedeau, Viola Bordunov, Chris Broka, Michelle F. Browner, Mario Cardozo, Peng Cheng, David Clark, Stacie Dalrymple, Michael DeGraffenreid, Adrian Gill, Xiaolin Hao, Ronald C. Hawley, Xiao He,