Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10591719 | Bioorganic & Medicinal Chemistry Letters | 2013 | 5 Pages |
Abstract
Structure guided optimization led to a potent series of JNK inhibitors with good physicochemical properties and desirable kinase selectivity as exemplified by compound 17.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Leyi Gong, Xiaochun Han, Tania Silva, Yun-Chou Tan, Bindu Goyal, Parch Tivitmahaisoon, Alejandra Trejo, Wylie Palmer, Heather Hogg, Alam Jahagir, Muzaffar Alam, Paul Wagner, Karin Stein, Lubov Filonova, Brad Loe, Ferenc Makra, David Rotstein,