Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10592102 | Bioorganic & Medicinal Chemistry Letters | 2014 | 4 Pages |
Abstract
Studies of the in vitro vascular properties of 4-(arylmethoxy)-1-alkylpiperidine inhibitors of the dopamine transporter are reported. The lipophilicity given by the size of the N-aryl substituent potentiated the inhibitory effect with 4a being the most effective blocker of KCl and noradrenaline-induced contractions.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Victor M. Pulgar, Jill Keith Harp,