Discovery of potent, reversible MetAP2 inhibitors via fragment based drug discovery and structure based drug design-Part 2

Article ID	Journal	Published Year	Pages	File Type
10592650	Bioorganic & Medicinal Chemistry Letters	2016	5 Pages	PDF

Keywords

FBDD SBDD MetAP2 Structure-based drug design Metalloprotease Fragment-based drug discovery

Related Topics

Physical Sciences and Engineering Chemistry Organic Chemistry

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Discovery of potent, reversible MetAP2 inhibitors via fragment based drug discovery and structure based drug design-Part 2

Authors

Christopher McBride, Zacharia Cheruvallath, Mallareddy Komandla, Mingnam Tang, Pamela Farrell, J. David Lawson, Darin Vanderpool, Yiqin Wu, Douglas R. Dougan, Artur Plonowski, Corine Holub, Chris Larson,