Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10593032 | Bioorganic & Medicinal Chemistry Letters | 2013 | 5 Pages |
Abstract
2-[(7-Nitrobenzo[c][1,2,5]oxadiazol-4-yl)thio]pyridine 1-oxide was identified as a potent inhibitor of KIX-KID interaction from screening the NCI diversity set. Further structure-activity relationship studies identified 4-aniline substituted nitrobenzofurazans with improved selectivity.
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Authors
Fuchun Xie, Bingbing X. Li, Candice Broussard, Xiangshu Xiao,