Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10593609 | Bioorganic & Medicinal Chemistry Letters | 2015 | 43 Pages |
Keywords
HMQCCPManti-silencing function 1IPTGDTTASF1H3K56acIC50GSHAstraZenecaREOsTFAH3K9UPLCSIRH3K27HRMSCOABMESARPBSFHTSPan-Assay Interference CompoundsH3K56MECNRtt109histone H3 lysine 27histone H3 lysine 9nuclear magnetic resonanceBSADMSODNAm/zSDS–PAGEβ-mercaptoethanolbovine serum albuminEDTAEthylenediaminetetraacetic acidAcetonitrileacetyl coenzyme AAcetyl-CoAdeoxyribonucleic acidTrifluoroacetic acidSodium dodecyl sulfate polyacrylamide gel electrophoresisheteronuclear multiple quantum coherenceisopropyl β-D-1-thiogalactopyranosideNMRPAINSdithiothreitolDimethyl sulfoxideStructure–activity relationshipStructure–activity relationshipsPartition coefficientDistribution coefficientMass spectrometryhigh-resolution mass spectrometryhigh-throughput screeningMethanolMeOHMass-to-charge ratiohalf maximal inhibitory concentrationHistone acetyltransferaseLog Dlog PUltra-performance liquid chromatographyHPLChigh-performance liquid chromatographyDrug discoveryHATcoenzyme AGlutathione
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Jayme L. Dahlin, J. Willem M. Nissink, Subhashree Francis, Jessica M. Strasser, Kristen John, Zhiguo Zhang, Michael A. Walters,