| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 10593805 | Bioorganic & Medicinal Chemistry Letters | 2012 | 6 Pages |
Abstract
A potent ghrelin receptor antagonist was discovered. The SAR studies around this structure and modifications to improve metabolic liabilities and rat PK are described.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Jeffrey T. Mihalic, Yong-Jae Kim, Mike Lizarzaburu, Xiaoqi Chen, Jeff Deignan, Malgorzata Wanska, Ming Yu, Jiasheng Fu, Xi Chen, Alex Zhang, Richard Connors, Lingming Liang, Michelle Lindstrom, Ji Ma, Liang Tang, Kang Dai, Leping Li,